Source: NORTH CAROLINA A&T STATE UNIV submitted to
CARNOSIC ACID ENRICHED ROSEMARY EXTRACT AND ITS ACTIVE COMPONENTS REDUCE WEIGHT GAIN AND TYPE 2 DIABETES
Sponsoring Institution
National Institute of Food and Agriculture
Project Status
TERMINATED
Funding Source
Reporting Frequency
Annual
Accession No.
0226277
Grant No.
2011-38821-31131
Project No.
NCE-2011-02447
Proposal No.
2011-02447
Multistate No.
(N/A)
Program Code
EQ
Project Start Date
Sep 1, 2011
Project End Date
Aug 31, 2014
Grant Year
2011
Project Director
Sang, S.
Recipient Organization
NORTH CAROLINA A&T STATE UNIV
1601 EAST MARKET STREET
GREENSBORO,NC 27411
Performing Department
(N/A)
Non Technical Summary
Within the last decade, obesity has increased dramatically on a global scale. Poor diet habit is one of the most common causes of excessive weight gain in today?s society and dietary intervention has been proven to be an effective approach to reduce the risk of obesity and related type 2 diabetes. We and others have found that rosemary extract has the antiobesity and antidiabetic effects. The objectives of this project are to identify the active components in rosemary extract and the effective dose of the active components and rosemary extract to reduce weight gain and type 2 diabetes in high-fat-fed mice, and to further understand the underlying molecular mechanisms. The development of this proposal is to build North Carolina A&T State University?s research capacity in the area of bioactive food components for prevention of obesity and related type 2 diabetes. New research activities created in this project will strengthen North Carolina A&T State University?s research capacity to study the beneficial health effects of functional foods and their bioactive components and to work with food industries to develop value-added functional foods to prevent chronic diseases, such as obesity and related type 2 diabetes.
Animal Health Component
(N/A)
Research Effort Categories
Basic
(N/A)
Applied
100%
Developmental
(N/A)
Classification

Knowledge Area (KA)Subject of Investigation (SOI)Field of Science (FOS)Percent
7021499101050%
7023840101050%
Goals / Objectives
The goals of this project are to identify the active components in rosemary extract and the effective dose of the active components and rosemary extract to reduce weight gain and type 2 diabetes in high-fat-fed mice, and to further understand the underlying molecular mechanisms. Our specific objectives are as follows: Objective 1. To determine the dose-dependent inhibitory effects of rosemary extract and its major components on obesity and type 2 diabetes in high-fat-fed mice by assessing a) Body weight and body fat gain b) Fasting blood glucose levels and plasma insulin levels c) Liver triglyceride levels Objective 2. Elucidate the mechanisms of inhibition of body weight gain and type 2 diabetes by rosemary extract and its active components in high-fat-fed mice. Using samples from Aim 1, we will examine the effects of the different treatments on a) Fecal lipids; b) Plasma inflammatory markers; c) Plasma leptin and adiponectin levels; d) Adipose tissue adiponectin and peroxisome-proliferator-activated-receptor (PPAR)-gamma levels. The expected ourputs from this project will be to observe inhibitory effects of carnosic acid enriched rosemary extract and its three major components, carnosic acid, carnosol and methoxy carnosic acid, on body weight and body fat gain and type 2 diabetes in high-fat-fed mice. We also expect to present our results at scientific meetings and publish them in peer-reviewed journals.
Project Methods
We will purify the three major components in rosemary extract for the proposed animal study in objective 1 and confirm their structures using MS and NMR. Then we will conduct the proposed animal study. We will recording the diet and body weight of the mice every week, and collecting fecal samples at 0, 5, 10, 12, 14, and 16 weeks of treatment. At 0, 5, 10, 12, 14, and 16 weeks of treatment, we will measure fasting blood glucose levels. After 16 weeks of treatment, we will sacrifice the mice and collect plasma and tissue samples for measurement of biomarkers discussed in Objective 2. For objective 2, we will identify the metabolites of the major components in rosemary extract and develop an LC/MS method to quantify their plasma and tissue levels. By accomplishing this project, we will present our results at scientific meetings and publish them in peer-reviewed journals. The accomplishment of stated objectives, results and measurable outcomes will be evaluated by the formed review committee focusing on the following questions: a) Does this project indeed build the research capacity of NCA&TSU b) Are students at NCA&TSU trained in this project as planned c) Is the proposed research conducted as planned

Progress 09/01/11 to 08/31/14

Outputs
Target Audience: The project's target audience included one graduate student, a post-doctorialcandidate as well as members of the general public who have metabolic syndrome. Changes/Problems: Nothing Reported What opportunities for training and professional development has the project provided? This project provided training of a graduate student and the thesis of this PhD student is part of the research of this project. How have the results been disseminated to communities of interest? Scientistsdisseminatedresults through scientific conferences.One student,Rashin Sedighi won the Nutraceutical and Functional Foods Division Poster Competition Award (First-Place) at the 2013 IFT annual meeting. What do you plan to do during the next reporting period to accomplish the goals? Nothing Reported

Impacts
What was accomplished under these goals? The major accomplishments of this project are: 1.Researchers developed a purification method to purify carnosic acid from rosemary extract and to prepare carnosic acid enriched rosemary extract in large quantities for the proposed mouse study using the combination of different types of column chromatography techniques. 2. Researchers identified carnosic acid as the major active component in rosemary extract to prevent the development of weight gain and metabolic syndrome induced by a high-fat diet in mice. 3. Researchers found that carnosic acid has a dose-dependent inhibitory effect against high-fat diet induced obesity and metabolic syndrome. 4. The potential underlying molecular mechanism is through inhibition of fat absorption by carnosic acid and rosemary extract. 5. Carnosic acid and rosemary extract could also attenuate oxidative stress, inflammation and formation of advanced glycation end products induced by a high-fat diet.

Publications

  • Type: Conference Papers and Presentations Status: Published Year Published: 2014 Citation: Carnosic acid as the major active component in rosemary ameliorates high-fat diet induced obesity and metabolic syndrome in mice
  • Type: Theses/Dissertations Status: Under Review Year Published: 2015 Citation: Carnosic Acid Enriched Rosemary Extract Inhibits Obesity and Metabolic Syndrome in High-fat-fed Mice


Progress 09/01/12 to 08/31/13

Outputs
Target Audience: Nothing Reported Changes/Problems: Nothing Reported What opportunities for training and professional development has the project provided? Nothing Reported How have the results been disseminated to communities of interest? Researchers gave one presentation at the 2013 IFT annual meeting. What do you plan to do during the next reporting period to accomplish the goals? Researchers plan to finish the proposed mouse study and analyze the samples collected from this study and also expect to publish at least one manuscript in the new fiscal year.

Impacts
What was accomplished under these goals? Researchers have prepared the carnosic acid-enriched rosemary extract for mouse study. The proposed mouse study is ongoing and is expecting to be finished by the end of 2013. The initial results indicate that rosemary extract and carnosic acid-enriched rosemary extract can inhibit body weight gain and fasting blood glucose levels.

Publications

  • Type: Conference Papers and Presentations Status: Published Year Published: 2013 Citation: Seldighi, R.; Chen, H.; Sang, S. Carnosic acid enriched rosemary extract inhibits obesity and metabolic syndrome in high-fat-fed mice. IFT Annual Meeting, Chicago, IL, July 13-16, 2013. (Poster)


Progress 09/01/11 to 08/31/12

Outputs
OUTPUTS: Obesity has reached epidemic proportions and remains the leading cause of preventable diseases including diet-related diabetes, heart disease, and hypertension. Dietary intervention has been proven to be an effective approach to reduce the risk of obesity and related type 2 diabetes. The goal of this project is to develop rosemary extract and its active components as cost-effective dietary strategies to prevent the development of obesity and related chronic diseases. We are training a graduate student at NCA&TSU to purify carnosic acid from rosemary extract. This student was also trained in terms of how to conduct a comprehensive literature search on the chemistry, bioavailability, and anti-obesity and anti-diabetic effects of rosemary extract and its active components. She was able to give a seminar entitled "Carnosic acid enriched rosemary extract and tis active components reduced weight gain and type 2 diabetes" to other graduate students and faculty at NCA&TSU. PARTICIPANTS: One graduate student, Mrs. Rashin Sedighi, is trained in this project. TARGET AUDIENCES: Nothing significant to report during this reporting period. PROJECT MODIFICATIONS: Nothing significant to report during this reporting period.

Impacts
We have successfully developed column chromatographic methods to purify carnosic acid and carnosol from rosemary extract. We are purifying carnosic acid in large quantify for the proposed mouse study.

Publications

  • No publications reported this period